Patents
Patents for A61K 31 - Medicinal preparations containing organic active ingredients (785,912)
04/2005
04/28/2005WO2005002522A3 Compositions and methods for treating tissue ischemia
04/28/2005WO2005002495A3 Use of plasma membrane calcium atpase (pmca) inhibitors for inhibiting sperm mobility
04/28/2005WO2005000282A3 Inhibitors of histone deacetylases for the suppression therapy of diseases
04/28/2005WO2005000243A3 The polymorphic form a of 4-[6-acetyl-3-[3-(4-acetyl-3-hydroxy-2-propylphenylthio)propoxy]-2-propylphenoxy]butryric acid
04/28/2005WO2005000232A3 Six membered amino-amide derivatives as angiogenesis inhibitors
04/28/2005WO2004110351A3 Heterocyclic compounds for treating hepatitis c virus
04/28/2005WO2004108682A3 Tetrahydroisoquinolines as antagonists of the 5ht1b receptor
04/28/2005WO2004108139A8 Use of fused heterocyclic compounds as scce inhibitors for the treatment of skin conditions or cancer
04/28/2005WO2004106299A3 Substituted pyrrole derivatives and their use as hmg-co inhibitors
04/28/2005WO2004099213A3 Pyrrolo (1,2-b) pyridazine compounds and their use as crf-1 receptor antagonists
04/28/2005WO2004098634A3 Protein arginine n-methyltransferase 2 (prmt-2)
04/28/2005WO2004098531A3 Increased transduction using abc transporter substrates and/or inhibitors
04/28/2005WO2004093817A3 Chemokine receptor binding heterocyclic compounds with enhanced efficacy
04/28/2005WO2004089293A3 Hydroxamic acid compounds and methods of use thereof
04/28/2005WO2004084905A3 Use of 5-ht2c receptor activity affecting compounds for treating idiopathic hyperhidrosis and associated conditions
04/28/2005WO2004075893A8 Method of treatment of cardiac and/or renal failure using a calcium channel blocker and an angiotensin converting enzyme inhibitor or an angiotensin ii receptor blocker
04/28/2005WO2004071437A3 Compositions for enhancing sexual responsiveness
04/28/2005WO2004065539A3 Androgen receptor antagonists
04/28/2005WO2004064759A3 Use of tryptanthrin compounds for immune potentiation
04/28/2005WO2004060378A8 Compositions comprising particles containing alumina with compounds bound to the alumina surface, delivery systems and methods of preparation thereof
04/28/2005WO2004050833A3 Glyceraldehyde 3-phosphate dehydrogenase-s(gapds), a glycolytic enzyme expressed only in male germ cells,is a target for male contraception
04/28/2005WO2004048524A3 Modulation of stat2 expression
04/28/2005WO2004035000A3 Enhancement of sleep with t-type calcium channel antagonists
04/28/2005WO2004014844A3 Aryl and heteroaryl compounds and methods to modulate coagulation
04/28/2005WO2004014842A8 Acylated arylcycloalkylamines and their use as pharmaceuticals
04/28/2005WO2004005262A8 New neuropeptide y y5 receptor antagonists
04/28/2005WO2003101425A8 Therapeutic agent-containing polymeric nanoarticles
04/28/2005WO2003099201A3 Compositions and methods of use for a fibroblast growth factor
04/28/2005WO2003095971A3 Posh nucleic acids, polypeptides and related methods
04/28/2005WO2003089597A3 Use of cox-2 inhibitors to prevent recurrences of herpesvirus infections
04/28/2005WO2003087389A3 Biologic modulations with nanoparticles
04/28/2005WO2003086283A9 Metastasis modulating activity of highly sulfated oligosaccharides
04/28/2005WO2003072067A3 Compositions and methods for treating epithelial and retinal tissue diseases
04/28/2005WO2003068929A3 Methods of inhibiting hiv-1 vpr activity and hiv-1 infectivity using atr or rad17 inhibitors
04/28/2005WO2003044170A3 Cyclic amp phosphodiesterase 4d7 isoforms and methods of use
04/28/2005US20050090752 Method for evaluating and treating hypertension
04/28/2005US20050090693 Clusianon derivatives; anticarcinogenic, antitumor and viricidal agents; mixture with mitogen-activated protein (MAP) kinase inhibitors
04/28/2005US20050090672 Intermediates for production of losartan; chloroformylation; hydroxylation; angiotensin II antagonists; hypertension
04/28/2005US20050090671 for human telomeres/telomerases; drug screening
04/28/2005US20050090669 Aminoalcohol derivatives as beta-3 adrenergic receptor agonists
04/28/2005US20050090661 For use as heat shock protein expression promoter, cell injury/death inhibitor, and cell and tissue protecting agent (organ preservation agent), antiulcer agent, antihepatopathic agent, and interleukin production promoter
04/28/2005US20050090564 Compositions and treatments of bacterial vaginosis
04/28/2005US20050090562 1-benzoyl-8,8-dimethyl-2-hydroxy-3,5,7-tris(3-methyl-2-butenyl)bicyclo- [3.3.]non-2-ene-4,9-dione and a protein kinase inhibitor; antineoplastic agents; antiproliferative agents
04/28/2005US20050090561 Cardiovascular disorders eg venous thrombosis, arterial thrombosis, deep vein thrombosis, pulmonary embolism, unstable angina, myocardial infarction, cardiac ischemia, occlusive diseases of the peripheral arteries and atrial fibrillation, smooth muscle cell proliferation, atherosclerosis, arteriosclerosi
04/28/2005US20050090558 Suppressing immune response in a mammal comprising accelerating lymphocyte homing (ALH) to any of mesenteric or peripheral lymph tissues or Peyer's patches by administering an ALH-immunosuppressive compound
04/28/2005US20050090557 Methods and compositions for administration of TRPV1 agonists
04/28/2005US20050090556 Method for treatment of external secretion disorders
04/28/2005US20050090555 Compound for the treatment of metabolic disorders
04/28/2005US20050090554 Administering baclofen, or a salt thereof, to relieve at least one symptom of gastroparesis other than vomiting
04/28/2005US20050090553 Compositions and method for treatment of chronic inflammatory diseases
04/28/2005US20050090552 Crystalline form with xray powder diffraction pattern peaks at 4.7, 7.4, 13.8 and 17.0+-0.2 but not at 3.8+-0.2 theta; thermal stability
04/28/2005US20050090551 Therapeutic use of methionine for the treatment or prevention of mucositis
04/28/2005US20050090550 Treating and/or preventing urinary incontinence using prodrugs of GABA analogs
04/28/2005US20050090549 Intrathecal gabapentin for treatment of pain
04/28/2005US20050090548 Intrathecal gabapentin for treatment of epilepsy
04/28/2005US20050090547 Combinations of retigabine and sodium channel inhibitors or sodium channel-influencing active compounds for treating pains
04/28/2005US20050090545 Nitric oxide topical technology
04/28/2005US20050090544 Oxaliplatin formulations
04/28/2005US20050090543 Method for the preparation of tetrahydrobenzothiepines
04/28/2005US20050090542 crystalline polymorphic dosage forms of anticholesterol agents; statins
04/28/2005US20050090541 Indolinone derivatives and their use in treating disease-states such as cancer
04/28/2005US20050090540 E.g., 2,2-bis(hydroxymethyl)-1 -azabicyclo[2,2,2]octan-3-one and 2-hydroxymethyl-3,3-dihydroxy-1-azabicyclo[2,2,2]octane; these compounds reactivate the apoptosis-inducing function of mutant p53 proteins and are used to treat various types of tumors
04/28/2005US20050090539 Intermediates for making 1(alpha-amino-1-(cyclopropyl-fused pyrrolidinylcarbonyl)methyl)-3-hydroxyadamantanes, e.g., methyl 3-hydroxy-<a-oxotricyclo[3.3.1.13,7]decane-1-acetate
04/28/2005US20050090538 Potentiating an NSAID and/or acetaminophen analgesic by administering concurrently a cyclooxygenase-2 inhibitor such as celecoxib, meloxicam, nimesulide and/or rofecoxib
04/28/2005US20050090537 Pharmaceutical composition based on idazoxan, salts, hydrates or polymorphs thereof
04/28/2005US20050090536 Substituted pyrrol-3-ylisoxazoles, e.g., N-benzyl-4-[4-(o-chlorophenyl)-5-isoxazolyl)pyrrole-2-carboxamide; treating diseases that are alleviated by a protein kinase inhibitor, particularly cancer, inflammatory disorders, restenosis, and cardiovascular disease.
04/28/2005US20050090535 Epothilones C, D, E and F, preparation and compositions
04/28/2005US20050090533 Treating schizophrenia by administering an N-(2-aminopyridin-5-yl)amino-phenylisobutyramide, e.g., N-[6-(2-acetylamino-ethylamino)-4-(2-chloro-phenyl)-pyridin-3-yl]-2-(3,5-bis-trifluoromethyl-phenyl)-N-methyl-isobutyramide
04/28/2005US20050090532 Medicinal uses of dihydropyrazoles
04/28/2005US20050090531 MAG expression promoters
04/28/2005US20050090530 5-(4-(2-(n-methyl-n-(2-pyridyl)amido)ethoxy)benzyl)thiazolidine-2, 4-dione and pharmaceutical compositions comprising the same
04/28/2005US20050090529 5-pyridin-3-yl-substituted, e.g., 5-(5-ethylaminomethyl-4-methylpyridin-3-yl)-3-(1H-imidazol-2-yl)-1H-indazole; CDK mediators, used to treat cancer, as well as proliferative diseases such as diabetic retinopathy, neovascular glaucoma, rheumatoid arthritis, and psoriasis
04/28/2005US20050090527 H1 antagonists used include loratadine, desloratadine, cetirizine and fexofenadine; H3 antagonists used include thioperamide, impromidine, burimamide, clobenpropit, impentamine, and mifetidine; and H4 antagonists used include dual H3/H4 antagonists
04/28/2005US20050090526 3-Cyano-7-methoxy-4-(3-bromo-4,5-dimethoxyphenyl)-2-oxo-2H-chromene; 7-Amino-4-(3-bromo-4,5-dimethoxy-phenyl)-3-cyano-2-imino-2H-chromene; anticancer, antitumor agent
04/28/2005US20050090525 carboxymethylated N-(nitrogen group functionalized alkyl- carbonylhydrazido)- or carbonylaminomethylcarbonyl)- substituted; integrin inhibitors used for combating thromboses, cardiac infarction, coronary heart diseases, arteriosclerosis, inflammation, tumors, osteoporosis, infections and restenosis
04/28/2005US20050090524 Novel adamantane derivatives
04/28/2005US20050090523 2-(substituted phenyl)imidazo[1,2-a]pyridine compounds; use to treat disorders mediated by the histamine H3 receptor such as sleep disorders, attention deficit hyperactivity disorder, or Alzheimer's disease; 2-[4-[3-(Piperidino)propylamino]phenyl]-8-methylimidazo[1,2-a]pyridine for example
04/28/2005US20050090521 Tetrazoloquinoline, triazoloquinoline, and oxazoloquinoline compounds, e.g., 9-chloro-N-isopropoxytetrazolo[1,5-a]quinoline-4-carboxamide
04/28/2005US20050090520 Treatment of disease or injury of the nervous system with FTY720
04/28/2005US20050090519 1-Alkyl-4-(3-substitutedphenyl)piperidines
04/28/2005US20050090518 Method for treating parkinson's disease using apomorphine and apomorphine prodrugs
04/28/2005US20050090517 Pharmaceutical combinations of cox-2 inhibitors and opiates
04/28/2005US20050090516 Novel substituted imides
04/28/2005US20050090515 anticarcinogenic, antitumor, antiproliferative agents; focal adhesion kinase (FAK) and cyclin-dependent kinase (CDK) enzyme inhibitors
04/28/2005US20050090514 Cool-genic compounds as anticarcinogenic agents promoting apoptosis and inhibit angiogenesis; antiproliferative agents
04/28/2005US20050090513 Compounds specific to adenosine a1 and a3 receptors and uses thereof
04/28/2005US20050090512 Method of treating extreme physical or mental stress using L-theanine to obtain accelerated regeneration
04/28/2005US20050090511 Synergistic combination of theanine and cystine for administration with foods, feeds, and beverages bases, confectioneries or powders; viricides, bactericides
04/28/2005US20050090510 Use of low molecular weight compounds for preparing a medicament useful in treating mutant p53 mediated diseases
04/28/2005US20050090507 Administered singly or in combination with a second antineoplastic agent; cyclin-dependent kinase inhibitors, antiproliferative agents; coupling and cyclization of a 1-aminopyridazinium salt with a 2-alkylthio-4-alkynyl pyrimidine compound
04/28/2005US20050090505 Methods of reducing risk of infection from pathogens
04/28/2005US20050090504 Crohn's disease, ulcerative colitis, asthma, hypersensitivity pneumonitis, eosinophilic pneumonias, rhinitis, psoriasis, dermatitis and eczema
04/28/2005US20050090503 5-HT receptor ligands and uses thereof
04/28/2005US20050090502 Protein tyrosine phosphatase 1B inhibitors alone or incombination with other antidiabetic, antilipemic, anticholesterol or hypotensive agents
04/28/2005US20050090501 Heteroaryl-cyclic acetals
04/28/2005US20050090500 Oral administration of a crystalline form of erlotinib hydrochloride to treat cancer expressing epidermal growth factor receptor (EGFR), including non-small cell lung cancer, head and neck cancer, or ovarian cancer
04/28/2005US20050090499 Oral or injectable dosage forms; antiproliferative, anticarcinogenic, and antiinflammatory agents; ATP hydrolysis inhibition
04/28/2005US20050090497 Novel ester or amide derivatives
04/28/2005US20050090496 Sulphonyl compounds with 5-ht6 receptor affinity
04/28/2005US20050090494 Such as N-[2-(3-{[1-(3,4-dichlorobenzylpiperidinyl]aminohydroxypropoxy)phenyl]acetamide; antiinflammatory agents, antiarthritic agents; chronic obstructive pulmonary disease, asthma, multiple sclerosis